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Polyethylenimine, an Autophagy-Inducing Platinum-Carbene-Based Drug Carrier with Potent Toxicity towards Glioblastoma Cancer Stem Cells.

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Red Light-Responsive Upconverting Nanoparticles for Quantitative and Controlled Release of a Coumarin-Based Prodrug.

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An N-heterocyclic carbene iridium(III) complex as a potent anti-cancer stem cell therapeutic.

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Polyarginine as a simultaneous antimicrobial, immunomodulatory and miRNA delivery agent within polyanionic hydrogels.

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Design of Oligourea-Based Foldamers with Antibacterial and Antifungal Activities.

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Design of a new cell penetrating peptide for DNA, siRNA and mRNA delivery.

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J Gene Med. 2021 Dec 2;:e3401

Different Biological Activities of Histidine-Rich Peptides Are Favored by Variations in Their Design.

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Delivery of siRNA by tailored cell-penetrating urea-based foldamers.

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Characterization of the DNA and Membrane Interactions of a Bioreducible Cell Penetrating Foldamer in Its Monomeric and Dimeric Form.

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Membrane pore-formation correlates with the hydrophilic angle of histidine-rich amphipathic peptides with multiple biological activities.

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Peptides derived from the C-terminal domain of HIV-1 Viral Protein R in lipid bilayers: Structure, membrane positioning and gene delivery.

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Biochim Biophys Acta Biomembr. 2019 Dec 6;:183149

Design and evaluation of ionizable peptide amphiphiles for siRNA delivery.

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Hybrid Cell-Penetrating Foldamer with Superior Intracellular Delivery Properties and Serum Stability.

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Bioconjug. Chem.. 2019 Apr 17;30(4):1133-1139

Induction of tumor-specific CTL responses using the C-terminal fragment of Viral protein R as cell penetrating peptide.

Gross DA, Leborgne C, Chappert P, Masurier C, Leboeuf M, Monteilhet V, Boutin S, Lemonnier FA, Davoust J, Kichler A

Sci Rep. 2019 Mar 8;9(1):3937

Cationic Photopolymerized Polydiacetylenic (PDA) Micelles for siRNA Delivery.

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Co-delivery of anti-PLK-1 siRNA and camptothecin by nanometric polydiacetylenic micelles results in a synergistic cell killing.

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RSC Adv. 2018 Jun 5;8(37):20758-20763

Polydiacetylenic nanofibers as new siRNA vehicles for in vitro and in vivo delivery.

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Nanoscale. 2018 Jan 25;10(4):1587-1590

The absorption enhancer sodium deoxycholate promotes high gene transfer in skeletal muscles.

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Histidine-rich designer peptides of the LAH4 family promote cell delivery of a multitude of cargo.

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J Control Release. 2017 Jan;246:60-70

pH-Responsive Nanometric Polydiacetylenic Micelles Allow for Efficient Intracellular siRNA Delivery.

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Molecular Determinants of Vectofusin-1 and Its Derivatives for the Enhancement of Lentivirally Mediated Gene Transfer into Hematopoietic Stem/Progenitor Cells.

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A Cell-Penetrating Foldamer with a Bioreducible Linkage for Intracellular Delivery of DNA.

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Efficient in vitro and in vivo pulmonary delivery of nucleic acid by carbon dot-based nanocarriers.

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Quantitative measurement of delivery and gene silencing activities of siRNA polyplexes containing pyridylthiourea-grafted polyethylenimines.

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Targeted gene transfer into hepatoma cells with lipopolyamine-condensed DNA particles presenting galactose ligands: a stage toward artificial viruses.

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