Dr BOURGUET Erika

Fiche personne

Coordonnées

Institut de Chimie Moléculaire de Reims
UMR CNRS 7312
51 rue Cognacq Jay
51096 REIMS Cedex

03 26 91 37 33

Territoire

Champagne-Ardenne

Statut

Enseignant-Chercheur

Affiliation

Université de Reims Champagne-Ardenne (URCA)

Institut de Chimie Moléculaire de Reims - UMR 7312 CNRS (ICMR)

Équipes/plateformes

UMR 7312 - Equipe "Biomolécules : Synthèse et Mécanismes d'Action (BSMA)"

Publications

Human Neuraminidases: Structures and Stereoselective Inhibitors.

Bourguet E, Figurska S, Fra Czek MM

J Med Chem. 2022 Feb 16;:

Targeting Class IIa HDACs: Insights from Phenotypes and Inhibitors.

Liu L, Dong L, Bourguet E, Fairlie DP

Curr Med Chem. 2021 Jun 29;:

How could histone deacetylase activators be useful leads in the search for new therapeutics?

Bourguet E, Naassila M

Future Med Chem. 2019 Jun 4;:

Unexpected effect of cyclodepsipeptides bearing a sulfonylhydrazide moiety towards histone deacetylase activity.

Létévé M, Gonzalez C, Moroy G, Martinez A, Jeanblanc J, Legastelois R, Naassila M, Sapi J, Bourguet E

Bioorg. Chem.. 2018 Aug 10;81:222-233

Interest of new alkylsulfonylhydrazide-type compound in the treatment of alcohol use disorders.

Jeanblanc J, Bourguet E, Sketriené D, Gonzalez C, Moroy G, Legastelois R, Létévé M, Trussardi-Régnier A, Naassila M

Psychopharmacology (Berl.). 2018 Apr 30;:

Class I HDAC Inhibitors: Potential New Epigenetic Therapeutics for Alcohol Use Disorder (AUD).

Bourguet E, Ozdarska K, Moroy G, Jeanblanc J, Naassila M

J. Med. Chem.. 2017 Aug;:

[Epigenetic mechanisms and alcohol use disorders: a potential therapeutic target].

Legastelois R, Jeanblanc J, Vilpoux C, Bourguet E, Naassila M

Biol Aujourdhui. 2017 ;211(1):83-91

Design, Synthesis, and Use of MMP-2 Inhibitor-Conjugated Quantum Dots in Functional Biochemical Assays.

Bourguet E, Brazhnik K, Sukhanova A, Moroy G, Brassart-Pasco S, Martin AP, Villena I, Bellon G, Sapi J, Nabiev I

Bioconjug. Chem.. 2016 Apr;27(4):1067-81

Neutrophil elastase as a target in lung cancer.

Moroy G, Alix AJ, Sapi J, Hornebeck W, Bourguet E

Anticancer Agents Med Chem. 2012 Jul;12(6):565-79.

Inhibition of human leukocyte elastase, plasmin and matrix metalloproteinases by oleic acid and oleoyl-galardin derivative(s).

Moroy G, Bourguet E, Decarme M, Sapi J, Alix AJ, Hornebeck W, Lorimier S

Biochem Pharmacol. 2011 Mar 1;81(5):626-35

The Total Synthesis of Trungapeptin A

Fecourt F, Sapi J, Bourguet E

Synlett. 2010 Feb;3:399-402

In silico study of MMP inhibition.

Rouffet M, Denhez C, Bourguet E, Bohr F, Guillaume D

Org Biomol Chem. 2009 Sep 21;7(18):3817-25

Control of Melanoma Invasiveness by Anticollagenolytic Agents: A Reappraisal of an Old Concept

Bourguet E, Sapi J, Emonard H, Hornebeck W

Anticancer Agents Med Chem. 2009 Jun;9(5):576-9.

Introduction of the 4-(4-bromophenyl)benzenesulfonyl group to hydrazide analogs of Ilomastat leads to potent gelatinase B (MMP-9) inhibitors with improved selectivity.

Ledour G, Moroy G, Rouffet M, Bourguet E, Guillaume D, Decarme M, Elmourabit H, Auge F, Alix AJ, Laronze JY, Bellon G, Hornebeck W, Sapi J

Bioorg Med Chem. 2008 Sep 15;16(18):8745-59

Looking forward: a glance into the future of organic chemistry.

Compain P, Desvergnes V, Ollivier C, Robert F, Suzenet F, Barboiu M, Belmont P, Bleriot Y, Bolze F, Bouquillon S, Bourguet E, Braida B, Constantieux T, Desaubry L, Dupont D, Stephane G, Jerome F, Legoupy S, Marat X, Marie M, Moitessier N, Papot S, Peri F, Petit M, Py S, Schulz E, Isabelle TO, Vauzeilles B, Philippe V, Vergnes L, Vidal S, Wilmouth S

New J Chem. 2006 Jun;30(6):823-31.

Future alchemy: account of the ESYOP experiment..

Compain P, Desvergnes V, Ollivier C, Robert F, Suzenet F, Barboiu M, Belmont P, Bleriot Y, Bolze F, Bouquillon S, Bourguet E, Braida B, Constantieux T, Desaubry L, Dupont D, Gastaldi S, Jerome F, Legoupy S, Marat X, Migaud M, Moitessier N, Papot S, Peri F, Petit M, Py S, Schulz E, Tranoy-Opalinski I, Vauzeilles B, Vayron P, Vergnes L, Vidal S, Wilmouth S

C R Chim. 2006 Jan;9(1):127-40.

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